The first enzymatic Achmatowicz reaction: selective laccase-catalyzed synthesis of 6-hydroxy-(2H)-pyran-3(6H)-ones and (2H)-pyran-2,5(6H)-diones
- Publication Type
- Journal contribution (peer reviewed)
- Authors
- Asta, C.; Schmidt, D.; Conrad, J.; Förster-Fromme, B.; Tolasch, T.; Beifuss, U.
- Year of publication
- 2013
- Published in
- RSC Adv.
- Band/Volume
- 3/
- DOI
- 10.1039/C3RA44107E
- Page (from - to)
- 19259-19263
The laccase-catalyzed oxidation of (5-alkylfuran-2-yl)carbinols using aerial oxygen as an oxidant selectively affords 6-hydroxy-(2H)-pyran-3(6H)-ones with yields up to 90%. With suitable substituted furan-2-yl carbinols as substrates the procedure allows the efficient preparation of (2H)-pyran-2,5(6H)-diones in a single step.